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Maja Kokot



Osebna bibliografija za obdobje 2013-2024





2013

1. KOKOT, Maja, KOSI, Danijel. Ozaveščenost ljudi o pomenu in varnosti jedrske energije : raziskovalna naloga. Ptuj: Gimnazija, 2013. 28 f., ilustr. [COBISS.SI-ID 24360504]


2019

2. KOKOT, Maja. Sinteza novih zaviralcev bakterijske DNA giraze A z 1,5-naftiridinskim skeletom = Synthesis of novel DNA Gyrase A inhibitors with 1,5-naphthyridine scaffold : enoviti magistrski študijski program Farmacija. Ljubljana: [M. Kokot], 2019. X, 54 f., ilustr. https://repozitorij.uni-lj.si/IzpisGradiva.php?id=109909. [COBISS.SI-ID 4785265]


2020

3. KROEZEN, Blijke S., CONTI, Gabriele, GIRARDI, Benedetta, CRAMER, Jonathan, JIANG, Xiaohua, RABBANI, Said, MÜLLER, Jennifer, KOKOT, Maja, LUISONI, Enrico, RICKLIN, Daniel, SCHWARDT, Oliver, ERNST, Beat. A potent mimetic of the Siglec-8 ligand 6ʹ-sulfo-sialyl ▫$Lewis^x$▫. ChemMedChem. 16 Sep. 2020, vol. 15, iss. 18, str. 1706-1719. ISSN 1860-7187. https://chemistry-europe.onlinelibrary.wiley.com/doi/epdf/10.1002/cmdc.202000417, DOI: 10.1002/cmdc.202000417. [COBISS.SI-ID 66592771]


2021

4. KOKOT, Maja. Breaking the wall of bacterial resistance. V: Falling Walls Lab : Science Summit 2021 : 7 Nov. 2021. [Berlin: s. n.; San Bruno]: YouTube [distributer], 2021. 1 spletni vir (1 videodatoteka (2 min 57 sek)). https://www.youtube.com/watch?v=qAc1SQ762oc. [COBISS.SI-ID 89042691]
5. KOLARIČ, Anja, KOKOT, Maja, HRAST, Martina, WEISS, Matjaž, ZDOVC, Irena, TRONTELJ, Jurij, ŽAKELJ, Simon, ANDERLUH, Marko, MINOVSKI, Nikola. A fine-tuned lipophilicity/hydrophilicity ratio governs antibacterial potency and selectivity of bifurcated halogen bond-forming NBTIs. Antibiotics. 2021, vol. 10, no. 7, art. 862, 30 str., ilustr., tabele. ISSN 2079-6382. https://www.mdpi.com/2079-6382/10/7/862, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.3390/antibiotics10070862. [COBISS.SI-ID 70416899]
projekt: P1-0017; financer: ARRS
projekt: P1-0208; financer: ARRS
6. KOKOT, Maja, MINOVSKI, Nikola. Prediction of binding affinity for combinatorially optimized NBTIs as Staphylococcus aureus and Escherichia coli DNA gyrase inhibitors by 6D-QSAR pseudoreceptor modeling. V: PINTAR, Albin (ur.), et al. Zbornik povzetkov = Book of abstracts : Slovenski kemijski dnevi 2021 = 27th Annual Meeting of the Slovenian Chemical Society : 22.-24. september 2021, Portorož, Portorose, Slovenija. Ljubljana: Slovensko kemijsko društvo, 2021. Str. 130. ISBN 978-961-93849-9-2. [COBISS.SI-ID 80589059]
7. KOKOT, Maja, WEISS, Matjaž, ZDOVC, Irena, HRAST, Martina, ANDERLUH, Marko, MINOVSKI, Nikola. Structurally optimized potent dual-targeting NBTI antibacterials with an enhanced bifurcated halogen-bonding propensity. ACS Medicinal Chemistry Letters. 2021, vol. 12, iss. 9, str. 1478-1485, ilustr. ISSN 1948-5875. https://pubs.acs.org/doi/10.1021/acsmedchemlett.1c00345, https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00345, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.1021/acsmedchemlett.1c00345. [COBISS.SI-ID 73185027]
projekt: P1-0017; financer: ARRS
projekt: P1-0208; financer: ARRS
projekt: 39010; financer: Young Researcher’s Program
8. KOKOT, Maja, WEISS, Matjaž, ZDOVC, Irena, HRAST, Martina, ANDERLUH, Marko, MINOVSKI, Nikola. Structurally optimized potent dual-targeting NBTI antibacterials with enhanced bifurcated halogen-bonding propensity. V: PINTAR, Albin (ur.), et al. Zbornik povzetkov = Book of abstracts : Slovenski kemijski dnevi 2021 = 27th Annual Meeting of the Slovenian Chemical Society : 22.-24. september 2021, Portorož, Portorose, Slovenija. Ljubljana: Slovensko kemijsko društvo, 2021. Str. 195. ISBN 978-961-93849-9-2. [COBISS.SI-ID 81082627]


2022

9. KOKOT, Maja, WEISS, Matjaž, ZDOVC, Irena, ANDERLUH, Marko, HRAST, Martina, MINOVSKI, Nikola. Diminishing hERG inhibitory activity of aminopiperidine-naphthyridine linked NBTI antibacterials by structural and physicochemical optimizations. Bioorganic chemistry. 2022, vol. 128, 14 str., ilustr. ISSN 0045-2068. https://www.sciencedirect.com/science/article/pii/S004520682200493X, DOI: 10.1016/j.bioorg.2022.106087. [COBISS.SI-ID 118137091]
projekt: P1-0017; financer: ARRS
projekt: P1-0208; financer: ARRS
10. KOKOT, Maja, WEISS, Matjaž, ZDOVC, Irena, ANDERLUH, Marko, HRAST, Martina, MINOVSKI, Nikola. Novel bacterial topoisomerase inhibitors with decreased hERG cardiotoxicity and retained antibacterial activity. V: PINTAR, Albin (ur.). Slovenski kemijski dnevi 2022 = 28th Annual Meeting of the Slovenian Chemical Society : zbornik povzetkov = book of abstracts : 21.-23. september 2022, Portorož, Portorose, Slovenija. Ljubljana: Slovensko kemijsko društvo, 2022. Str. 171. ISBN 978-961-95922-1-2. [COBISS.SI-ID 125103107]
11. KOKOT, Maja, MINOVSKI, Nikola, ANDERLUH, Marko, HRAST, Martina. Novel dual bacterial topoisomerases inhibitors with broadspectrum antibacterial activity. V: ESCMID/ASM Conference on Drug Development : meet the challenge of antimicrobial resistance. ESCMID/ASM Conference on Drug Development, October 4 – 7, 2022 Dublin, Ireland. [S. l.]: [s. n.], 2022. 1 str. https://www.escmid.org/login?ReturnTo=https%3A%2F%2Felibrary.escmid.org%2Fsaml%2Flogin%3FreturnTo%3D%2F%3Fsearch%25255Bquery%25255D%253D%252522ESCMID%2FASM%252520Conference%252520on%252520Drug%252520Development%252520%2525E2%252580%252593%252520Meet%252520the%252520Challenge%252520of%252520Antimicrobial%252520Resistance%252522%2526tab%253Ddocs%2523results. [COBISS.SI-ID 128228099]
12. HRAST, Martina, KOKOT, Maja, MINOVSKI, Nikola, ZDOVC, Irena, ANDERLUH, Marko. Razvoj novih zaviralcev bakterijskih topoizomeraz, učinkovitih proti večkratno odpornim bakterijam. Mikrobiolog.si. 2022, letn. 2, št. 2, str. 15-22, ilustr. ISSN 2784-4463. http://www.smd.si/publikacije/. [COBISS.SI-ID 133900803]
13. KOKOT, Maja, ANDERLUH, Marko, HRAST, Martina, MINOVSKI, Nikola. The structural features of novel bacterial topoisomerase inhibitors that define their activity on topoisomerase IV. Journal of medicinal chemistry. 2022, vol. 65, iss. 9, str. 6431–6440, ilustr. ISSN 0022-2623. https://pubs.acs.org/doi/10.1021/acs.jmedchem.2c00039, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.1021/acs.jmedchem.2c00039. [COBISS.SI-ID 106691587]
14. KOKOT, Maja, WEISS, Matjaž, ZDOVC, Irena, ANDERLUH, Marko, HRAST, Martina, MINOVSKI, Nikola. Tetrahydropyran and cyclohexane linked novel bacterial topoisomerase inhibitors with improved balanced antibacterial activity and safety profile. V: Book of abstracts : XXVII National meeting on medicinal chemistry : NPCF14 : 14th Young medicinal chemistsʼ symposium : Nuove prospettive in chimica farmaceutica : Università degli studi di Bari Aldo Moro, September 11-14, 2022. [Bari: Società di Chimica Italiana: Università degli studi di Bari Aldo Moro], 2022. Str. 76, ilustr. [COBISS.SI-ID 123655427]


2023

15. KOKOT, Maja, WEISS, Matjaž, ZDOVC, Irena, ŠENEROVIĆ, L., RADAKOVIC, Natasa, ANDERLUH, Marko, MINOVSKI, Nikola, HRAST, Martina. Amide containing NBTI antibacterials with reduced hERG inhibition, retained antimicrobial activity against gram-positive bacteria and in vivo efficacy. European journal of medicinal chemistry. [Print ed.]. 2023, vol. 250, str. 1-13, ilustr. ISSN 0223-5234. https://www.sciencedirect.com/science/article/pii/S0223523423000752, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.1016/j.ejmech.2023.115160. [COBISS.SI-ID 141418755]
projekt: P1-0017; financer: ARRS
projekt: P1-0208; financer: ARRS
projekt: 39010
projekt: 50503 Young researcher’s program
16. KOKOT, Maja, NOVAK, Doroteja, ZDOVC, Irena, ANDERLUH, Marko, HRAST, Martina, MINOVSKI, Nikola. Exploring alternative pathways to target bacterial type II topoisomerases using NBTI antibacterials: beyond halogen-bonding interactions. Antibiotics. 2023, vol. 12, no. 5, art. 930, str. 1-15, ilustr. ISSN 2079-6382. https://www.mdpi.com/2079-6382/12/5/930, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.3390/antibiotics12050930. [COBISS.SI-ID 153123075]


2024

17. KOKOT, Maja, MINOVSKI, Nikola. Dynamic profiling and binding affinity prediction of NBTI antibacterials against DNA gyrase enzyme by multidimensional machine learning and molecular dynamics simulations. ACS omega. Apr. 11, 2024, vol. 9, iss. 16, str. 18278–18295, ilustr. ISSN 2470-1343. https://pubs.acs.org/doi/10.1021/acsomega.4c00036, DiRROS - Digitalni repozitorij raziskovalnih organizacij Slovenije, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.1021/acsomega.4c00036. [COBISS.SI-ID 192354563]
18. ZORMAN, Maša, HRAST, Martina, KOKOT, Maja, MINOVSKI, Nikola, ANDERLUH, Marko. The overview of development of novel bacterial topoisomerase inhibitors effective against multidrug-resistant bacteria in an academic environment : from early hits to in vivo active antibacterials. European Journal of Pharmaceutical Sciences. [Print ed.]. 2024, vol. 192, 7 str., ilustr. ISSN 0928-0987. https://www.sciencedirect.com/science/article/pii/S0928098723002622, DOI: 10.1016/j.ejps.2023.106632. [COBISS.SI-ID 171802883]
19. KOKOT, Maja. Strukturno podprto načrtovanje in optimizacija selektivne toksičnosti novih zaviralcev bakterijske topoizomeraze tipa II = Structure-based design and optimization of selective toxicity of the novel bacterial topoisomerase type II inhibitors : doktorska disertacija. Ljubljana: [M. Kokot], 2024. 155 f., graf. prikazi, ilustr. [COBISS.SI-ID 189473795]



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