Roland J. Pieters

1. ERJAVEC, Bibi. Sinteza iminosladkornih gradnikov za multivalentno inhibicijo glikozidaz : diplomska naloga. Ljubljana: [B. Erjavec], 2015. 33 f., ilustr. [COBISS.SI-ID 1536497859]

2. ŠROT, Luka. Guanidinium iminosugar derivatives as precursors to Beta-glucocerebrosidase inhibitors = Gvanidino iminosaharidni derivati kot prekurzorji zaviralcev beta-glukocerebrozidaze. Ljubljana: [L. Šrot], 2017. V, 59 str., tabele, ilustr. http://www.ffa.uni-lj.si/docs/default-source/knjiznica-doc/magistrske/2017/srot_luka_mag_nal_2017.pdf?sfvrsn=2, Repository of the University of Ljubljana – RUL . [COBISS.SI-ID 4429681]

3. SHI, Jie, TOMAŠIČ, Tihomir, SHARIF, Suhela, BROUWER, Arwin J., ANDERLUH, Marko, RUIJTENBEEK, Rob, PIETERS, Roland J. Peptide microarray analysis of the cross-talk between O-GlcNAcylation and tyrosine phosphorylation. FEBS letters. 2017, vol. 591, iss. 13, str. 1872-1883, ilustr. ISSN 1873-3468. http://onlinelibrary.wiley.com/doi/10.1002/1873-3468.12708/full, DOI: 10.1002/1873-3468.12708. [COBISS.SI-ID 4336753]
project: P1-0208; funder: ARRS
project: 20130618006; funder: China Scholarship Council

4. RUGEL, Maša. Sinteza gvanidinskih iminosladkorjev kot prekurzorjev za nove selektivne zaviralce beta - glukozidaze = Synthesis of guanidinlated iminosugars as precursors for new selective beta - glucosidase inhibitors : Uniform master's programme Pharmacy. Ljubljana: [M. Rugel], 2017. IX, 71 f., A - W f. pril., ilustr. http://www.ffa.uni-lj.si/docs/default-source/knjiznica-doc/magistrske/2017/rugel_masa_mag_nal_2017.pdf?sfvrsn=2, Repository of the University of Ljubljana – RUL . [COBISS.SI-ID 4417649]

5. RIHTER, Jakob. Sinteza iminosladkornih zaviralcev glukocerebrozidaze beta = Synthesis of iminosugar beta glucocerebrosidase inhibitors : enoviti magistrski študij farmacije. Ljubljana: [J. Rihter], 2017. X, 51 f., ilustr. http://www.ffa.uni-lj.si/docs/default-source/knjiznica-doc/magistrske/2017/rihter_jakob_mag_nal_2017.pdf?sfvrsn=2, Repository of the University of Ljubljana – RUL . [COBISS.SI-ID 4408433]

6. WEISS, Matjaž, TOMAŠIČ, Tihomir, ZHANG, Hao, SHI, Jie, RUIJTENBEEK, Rob, PIETERS, Roland J., ANDERLUH, Marko. Fragment based design of O-GlcNAc transferase inhibitors. In: Book of abstracts. 5th EMFC Young Medicinal Chemist Symposium, September 6 -7, 2018, Ljubljana, Slovenia. Ljubljana: Slovensko farmacevtsko društvo, 2018. Str. 80, p023. https://drive.google.com/file/d/1shXK1I7rFzkKhyBgfifZWCSH0lAJxiK0/view. [COBISS.SI-ID 4589425]

7. WEISS, Matjaž, TOMAŠIČ, Tihomir, ZHANG, Hao, SHI, Jie, RUIJTENBEEK, Rob, PIETERS, Roland J., ANDERLUH, Marko. Fragment based design of O-GlcNAc transferase inhibitors. In: ANDERLUH, Marko (ed.). Book of abstracts. XXV International Symposium on Medicinal Chemistry, Ljubljana, Slovenia, September 2 - 6, 2018. Ljubljana: Slovensko farmacevtsko društvo, 2018. Str. 346, p425. [COBISS.SI-ID 4584817]

8. ZHAO, Han, TOMAŠIČ, Tihomir, SHI, Jie, WEISS, Matjaž, RUIJTENBEEK, Rob, ANDERLUH, Marko, PIETERS, Roland J. Inhibition of O-GlcNAc transferase (OGT) by peptidic hybrids. MedChemComm. 2018, vol. 9, iss. 5, str. 883-887, ilustr. ISSN 2040-2503. http://pubs.rsc.org/en/Content/ArticleLanding/2018/MD/C8MD00115D#!divAbstract, DOI: 10.1039/C8MD00115D. [COBISS.SI-ID 4494449]
project: P1-0208; funder: ARRS
project: 201306210049; funder: China Scholarship Council

9. SLUGA, Janja, TOMAŠIČ, Tihomir, BAJC, Gregor, HRAST RAMBAHER, Martina, ANDERLUH, Marko, PINTAR, Sara, TURK, Dušan, PIETERS, Roland J., NOVIČ, Marjana. Discovery of iminosugars as inhibitors of bacterial N-acetylglucosaminidase with potential antibacterial activity. In: EUROPIN Summer School on Drug Design, Vienna, 15-20. 9. 2019. Vienna: [s. n.]. 2019, str. [1-2]. https://moodle.univie.ac.at/mod/folder/view.php?id=3282537. [COBISS.SI-ID 40234757]

10. SHI, Jie, SHARIF, Suhela, BALSOLLIER, Cyril, RUIJTENBEEK, Rob, PIETERS, Roland J., JONGKEES, Seino A.K. C-Terminal tag location hampers in vitro profiling of OGT peptide substrates by mRNA display. ChemBioChem. 2020, vol. 22, iss. 4, str. 666-671, ilustr. ISSN 1439-7633. https://chemistry-europe.onlinelibrary.wiley.com/doi/10.1002/cbic.202000624, DOI: 10.1002/cbic.202000624. [COBISS.SI-ID 87285763]

11. BRICELJ, Aleša, LOI, Elena Maria, GOBEC, Martina, STEINEBACH, Christian, GÜTSCHOW, Michael, PIETERS, Roland J., SOSIČ, Izidor, ANDERLUH, Marko. Development of OSMI-4-based biochemical probes for OGT. In: Book of abstracts : 2nd Alpine Winter Conference on Medicinal and Synthetic Chemistry, St. Anton, Austria, 19 - 23, 2020. [S. l.: s. n.], 2020. Str. 94, ilustr. https://www.alpinewinterconference.org/v2/data/1579181858BookAbstracts-Web.pdf. [COBISS.SI-ID 4875377]

12. SLUGA, Janja, TOMAŠIČ, Tihomir, BAJC, Gregor, HRAST RAMBAHER, Martina, ANDERLUH, Marko, PINTAR, Sara, TURK, Dušan, PIETERS, Roland J., NOVIČ, Marjana. Iminosugars as inhibitors of Staphylococcus aureus N-acetylglucosaminidase with potential antibacterial activity. In: PINTAR, Albin (ed.), et al. Zbornik povzetkov = Book of abstracts : Slovenski kemijski dnevi 2020 = 26th Annual Meeting of the Slovenian Chemical Society : 16.-18. september 2020, Portorož, Portorose, Slovenija. Ljubljana: Slovensko kemijsko društvo, 2020. Str. 150. ISBN 978-961-93849-7-8. [COBISS.SI-ID 31323395]

13. LOI, Elena Maria, WEISS, Matjaž, PAJK, Stane, GOBEC, Martina, TOMAŠIČ, Tihomir, PIETERS, Roland J., ANDERLUH, Marko. Intracellular hydrolysis of small-molecule O-linked N-acetylglucosamine transferase inhibitors differs among cells and is not required for its inhibition. Molecules. 2020, vol. 25, iss. 15, art. 3381, 10 str., ilustr. ISSN 1420-3049. https://www.mdpi.com/1420-3049/25/15/3381, Repository of the University of Ljubljana – RUL , DOI: 10.3390/molecules25153381. [COBISS.SI-ID 24851459]
project: 765581 PhD4GlycoDrug; funder: European Union’s Horizon2020 program under the Marie Skłodowska-Curie
project: CA18103 Innogly; funder: COST actions
project: CA18132 GLYCONanoPROBES; funder: COST Actions

14. LOI, Elena Maria, WEISS, Matjaž, BALSOLLIER, Cyril, TOMAŠIČ, Tihomir, PIETERS, Roland J., ANDERLUH, Marko. Different drug design approaches to tackle o-glcnac transferase inhibition. In: Book of abstracts. 2021. Str. 156, a009. https://www.efmc-ismc.org/v2/data/1630081893EFMC-ISMC-BookOfAbstracts-webHD.pdf. [COBISS.SI-ID 74924803]

15. WEISS, Matjaž, LOI, Elena Maria, STERLE, Maša, BALSOLLIER, Cyril, TOMAŠIČ, Tihomir, PIETERS, Roland J., GOBEC, Martina, ANDERLUH, Marko. New quinolinone O-GlcNAc transferase inhibitors based on fragment growth. Frontiers in chemistry. [Online ed.]. 2021, vol. 9, str. 1-8. ISSN 2296-2646. https://www.frontiersin.org/articles/10.3389/fchem.2021.666122/full, Repository of the University of Ljubljana – RUL , DOI: 10.3389/fchem.2021.666122. [COBISS.SI-ID 55702275]
project: P1-0208 Farmacevtska kemija: načrtovanje, sinteza in vrednotenje učinkovin; funder: ARRS
project: 765581 PhD4GlycoDrug; www.phd4glycodrug.eu; funder: European Union’s Horizon2020 programme under the Marie Skłodowska-Curie

16. BALSOLLIER, Cyril, PIETERS, Roland J., ANDERLUH, Marko. Overview of the assays to probe O-linked β-N-acetylglucosamine transferase binding and activity. Molecules. 2021, vol. 26, iss. 4, str. 1-20, ilustr. ISSN 1420-3049. https://www.mdpi.com/1420-3049/26/4/1037, Repository of the University of Ljubljana – RUL , DOI: 10.3390/molecules26041037. [COBISS.SI-ID 51829507]

17. SOSIČ, Izidor, STEINEBACH, Christian, BRICELJ, Aleša, NG, Y.L.D., GOBEC, Martina, KRÖNKE, Jan, PIETERS, Roland J., ANDERLUH, Marko, GÜTSCHOW, Michael. PROTACS as tools for the modulation of pharmacological targets : presented at early bird sessions on 45th FEBS Congress, Molecules of Life: Towards New Horizons, Ljubljana, Slovenia, July 3-8, 2021. FEBS open bio. 2021, vol. 11, suppl. s1, str. 100. ISSN 2211-5463. https://febs.onlinelibrary.wiley.com/doi/epdf/10.1002/2211-5463.13206, DOI: 10.1002/2211-5463.13206. [COBISS.SI-ID 70178051]

18. LOI, Elena Maria, TOMAŠIČ, Tihomir, BALSOLLIER, Cyril, VAN EEKELEN, Kevin, WEISS, Matjaž, GOBEC, Martina, ALTEEN, Matthew G., VOCADLO, David J., PIETERS, Roland J., ANDERLUH, Marko. Discovery of a new drug-like series of OGT inhibitors by virtual screening. Molecules. 2022, vol. 27, iss. 6, str. 1-21, tabele. ISSN 1420-3049. https://www.mdpi.com/1420-3049/27/6/1996, Repository of the University of Ljubljana – RUL , DOI: 10.3390/molecules27061996. [COBISS.SI-ID 101699843]
project: P1-0208; funder: ARRS
project: 765581; funder: European Union’s Horizon2020

19. ANDERLUH, Marko, LOI, Elena Maria, WEISS, Matjaž, BALLSOLIER, Cyril, TOMAŠIČ, Tihomir, GOBEC, Martina, PIETERS, Roland J. Inhibition of O-GlcNAc transferase - the cell's metabolic gauge that alters its fate : keynote lecture at the 15BSS Bratislava Symposium on Saccharides, June 20-24, 2022, Smolenice, Slovakia. https://www.saccharides.sav.sk/15BBS_programme.pdf. [COBISS.SI-ID 149551363]

20. LOI, Elena Maria, WEISS, Matjaž, PAJK, Stane, YASINI, Daniel, NOVAK, Doroteja, GOBEC, Martina, TOMAŠIČ, Tihomir, PIETERS, Roland J., ANDERLUH, Marko. The quest for the first potent in vivo acting OGT inhibitor. In: Book of abstracts. [S. l.]: [s. n.], 2022. Str. 152, p067. https://www.efmc-ismc.org/v2/data/1661849465EFMC-ISMC-Book-Web-HD3.pdf. [COBISS.SI-ID 121078275]

21. BALSOLLIER, Cyril, TOMAŠIČ, Tihomir, YASINI, Daniel, BIJKERK, Simon, ANDERLUH, Marko, PIETERS, Roland J. Design of OSMI-4 analogs using scaffold hopping : investigating the importance of the uridine mimic in the binding of OGT inhibitors. ChemMedChem. 2023, vol. 18, iss. 8, str. 1-7, ilustr. ISSN 1860-7187. https://chemistry-europe.onlinelibrary.wiley.com/doi/10.1002/cmdc.202300001, DOI: 10.1002/cmdc.202300001. [COBISS.SI-ID 141476867]
project: 765581 PhD4Glyco-Drug Innovative Training Network; funder: European Union’s Horizon 2020 research and innovation program under the Marie Skłodowska-Curie

22. LOI, Elena Maria. Structure-based design, synthesis and biological evaluation of novel O-β-N-acetylglucosaminyltransferase inhibitors = Strukturno podprto načrtovanje, sinteza in biološko vrednotenje novih zaviralcev O-β-N-acetilglukozaminil transferaze : interdisciplinary doctoral programme in biomedicine (Pharmacy) PhD programme in drug Innovation : doctoral dissertation. Ljubljana: [L. Elena Maria], 2023. 185 str., ilustr., graf. prikazi. Repository of the University of Ljubljana – RUL , http://www.dlib.si/details/URN:NBN:SI:doc-CDN2PGNO. [COBISS.SI-ID 146223619]

23. BALSOLLIER, Cyril, BIJKERK, Simon, DE SMIT, Arjen, VAN EKELEN, Kevin, BOZOVIČAR, Krištof, HUSSTEGE, Dirk, TOMAŠIČ, Tihomir, ANDERLUH, Marko, PIETERS, Roland J. Discovery of two non-UDP-mimic inhibitors of O-GlcNAc transferase by screening a DNA-encoded library. Bioorganic chemistry. 2024, vol. 147, str. 1-10, ilustr. ISSN 0045-2068. https://www.sciencedirect.com/science/article/pii/S0045206824002268, DOI: 10.1016/j.bioorg.2024.107321. [COBISS.SI-ID 191274499]
project: This work has been funded by the European Union’s Horizon 2020 research and innovation programme under the Marie Skłodowska Curie grant agreement No 765581 (PhD4GlycoDrug Innovative Training Network). The DELopen library and the off-DNA synthesis of hits were provided by WuXi AppTec.

24. SLUGA, Janja, TOMAŠIČ, Tihomir, ANDERLUH, Marko, HRAST RAMBAHER, Martina, BAJC, Gregor, SEVŠEK, Alen, MARTIN, Nathaniel I., PIETERS, Roland J., NOVIČ, Marjana, VENKO, Katja. Targeting N-acetylglucosaminidase in Staphylococcus aureus with iminosugar inhibitors. Antibiotics. 2024, vol. 13, iss. 8, [article no.] 751, str. 1-12, ilustr. ISSN 2079-6382. https://www.mdpi.com/2079-6382/13/8/751, Repository of the University of Ljubljana – RUL , DOI: 10.3390/antibiotics13080751. [COBISS.SI-ID 204113923]
project: This research was funded by the Slovenian Research and Inovation Agency (Grants P1-0017 and young researcher’s fund 39008).

25. BALSOLLIER, Cyril. The use of biological and computational tools to design, screen and synthesize new potent inhibitors of β-N-acetylglucosaminyl transferase = Uporaba bioloških in računalniških orodij za načrtovanje, testiranje in sintezo novih zaviralcev β-Nacetilglukozaminil transferaze : doctoral dissertation. Ljubljana: [C. Balsollier], 2024. 144 f., graf. prikazi. [COBISS.SI-ID 192124163]
project: 765581 project PhD4GlycoDrug; funder: European Union’s Horizon 2020 programme under the Marie Skłodowska-Curie