Jacques-Philippe Colletier

1. STOJAN, Jure, BROCHIER, Laure, ALIES, Carole, COLLETIER, Jacques-Philippe, FOURNIER, Didier. Inhibition of Drosophila melanogaster acetylcholinesterase by high concentations of substrate. European journal of biochemistry. 2004, letn. 271, str. 1364-1371. ISSN 0014-2956. [COBISS.SI-ID 19036633]

2. COLLETIER, Jacques-Philippe, FOURNIER, Didier, GREENBLATT, Harry M., STOJAN, Jure, SUSSMAN, Joel, ZACCAI, Giuseppe, SILMAN, Israel, WEIK, Martin. Structural insights into substrate traffic and inhibition in acetylcholinesterase. The EMBO journal. 2006, letn. 25, št. 12, str. 2746-2756. ISSN 0261-4189. [COBISS.SI-ID 21911001]

3. FRASCO, M.F., COLLETIER, Jacques-Philippe, WEIK, Martin, CARVALHO, Felix, GUILHERMINO, L., STOJAN, Jure, FOURNIER, Didier. Mechanisms of cholinesterase inhibition by inorganic mercury. FEBS journal. 2007, letn. 274, št. 7, str. 1849-1861. ISSN 1742-464X. [COBISS.SI-ID 22772185]

4. BRUS, Boris, KOŠAK, Urban, TURK, Samo, PIŠLAR, Anja, COQUELLE, Nicolas, KOS, Janko, STOJAN, Jure, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Discovery, biological evaluation, and crystal structure of a novel nanomolar selective butyrylcholinesterase inhibitor : [kratko predavanje]. In: ANDERLUH, Gregor (ed.), KRAŠEVEC, Nada (ed.). Molekulske interakcije : 10 let Infrastrukturnega centra za raziskave molekulskih interakcij : mini simpozij 2014, 3. 12. 2014, Ljubljana. Ljubljana: Laboratorij za molekularno biologijo in nanobiotehnologijo, Kemijski inštitut, 2014. Str. 28, ilustr. ISBN 978-961-6104-27-2. [COBISS.SI-ID 3786609]

5. BRUS, Boris, KOŠAK, Urban, TURK, Samo, PIŠLAR, Anja, COQUELLE, Nicolas, KOS, Janko, STOJAN, Jure, COLLETIER, Jacques-Philippe, GOBEC, Stanislav, et al. Discovery, biological evaluation, and crystal structure of a novel nanomolar selective butyrylcholinesterase inhibitor. Journal of medicinal chemistry. 2014, vol. 57, issue 19, str. 8167-8179, ilustr. ISSN 0022-2623. http://pubs.acs.org/action/doSearch?text1=Discovery%2C+Biological+Evaluation%2C+and+Crystal+Structure+of+a+Novel+Nanomolar+Selective+Butyrylcholinesterase+Inhibitor&field1=Title, http://pubs.acs.org/doi/pdf/10.1021/jm501195e, DOI: 10.1021/jm501195e. [COBISS.SI-ID 3713393]

6. BRUS, Boris, KOŠAK, Urban, KNEZ, Damijan, COQUELLE, Nicolas, ŽIVIN, Marko, SALAT, Kinga, PODKOWA, Adrian, FILIPEK, Barbara, WIĘCKOWSKA, Anna, MALAWSKA, Barbara, STOJAN, Jure, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Discovery of nanomolar inhibitors of butyrycholinesterase. In: IXthe Joint Meeting in Medicinal Chemistry, 7-10 June 2015, Athens, Greece : program. Athens: [s. n.], 2015. 1 str. http://www.efmc.info/infos.php?langue=english&cle_menus=1201086332&cle_data=1417004654. [COBISS.SI-ID 3997553]

7. KNEZ, Damijan, BRUS, Boris, COQUELLE, Nicolas, SOSIČ, Izidor, ŠINK, Roman, BRAZZOLOTTO, Xavier, MRAVLJAK, Janez, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Structure-based development of nitroxoline derivatives as potential multifunctional anti-Alzheimer agents. Bioorganic & Medicinal Chemistry. [Print ed.]. Aug. 2015, vol. 23, iss. 15, str. 4442-4452, ilustr. ISSN 0968-0896. http://www.sciencedirect.com/science/article/pii/S0968089615005040#, DOI: 10.1016/j.bmc.2015.06.010. [COBISS.SI-ID 3874161]

8. BRUS, Boris, KOŠAK, Urban, KNEZ, Damijan, COQUELLE, Nicolas, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. 1,3- in 1,4-disubstituirani piperidini kot zaviralci butirilholin-esteraze za zdravljenje Alzheimerjeve bolezni in ostalih demenc : 24951 (A), 2016-09-30. Ljubljana: Urad Republike Slovenije za intelektualno lastnino, 2016. 50 str., ilustr. http://www2.uil-sipo.si/ds1.htm?A=107000&Q=NUM%3D201500076. [COBISS.SI-ID 4223857]
patent family: Številka prijave: 201500076; Številka patenta: 24951 (A), 2016-09-30

9. KOŠAK, Urban, BRUS, Boris, KNEZ, Damijan, ŠINK, Roman, ŽAKELJ, Simon, TRONTELJ, Jurij, PIŠLAR, Anja, ŠLENC, Jasna, GOBEC, Martina, ŽIVIN, Marko, TRATNJEK, Larisa, PERŠE, Martina, SAŁAT, Kinga, PODKOWA, Adrian, FILIPEK, Barbara, NACHON, Florian, BRAZZOLOTTO, Xavier, WIĘCKOWSKA, Anna, MALAWSKA, Barbara, STOJAN, Jure, MLINARIČ-RAŠČAN, Irena, KOS, Janko, COQUELLE, Nicolas, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Development of an in-vivo active reversible butyrylcholinesterase inhibitor. Scientific reports. Dec.. 2016, vol. 6, str. 1-16, ilustr. ISSN 2045-2322. http://www.nature.com/articles/srep39495, DOI: 10.1038/srep39495. [COBISS.SI-ID 4263537]

10. KOŠAK, Urban, KNEZ, Damijan, BRUS, Boris, PIŠLAR, Anja, ŽAKELJ, Simon, TRONTELJ, Jurij, STOJAN, Jure, ŽIVIN, Marko, PODKOWA, Adrian, SAŁAT, Kinga, COQUELLE, Nicolas, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Development of in vivo active non - covalent butyrycholinesterase inhibitors. In: KLJUN, Jakob (ed.), GABER, Aljaž (ed.). Book of abstracts. Scientific Conference for Young Researchers, 19. 9. 2017. Ljubljana: Fakulteta za kemijo in kemijsko tehnologijo, 2017. Str. 10, ilustr. ISBN 978-961-6756-83-9. [COBISS.SI-ID 4405105]

11. KOŠAK, Urban, KNEZ, Damijan, COQUELLE, Nicolas, BRUS, Boris, PIŠLAR, Anja, NACHON, Florian, BRAZZOLOTTO, Xavier, KOS, Janko, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. N-propargylpiperidines with naphthalene-2-carboxamide or naphthalene-2- sulfonamide moieties. Bioorganic & Medicinal Chemistry. [Print ed.]. 2017, vol. 25, iss. 2, str. 633-645, ilustr. ISSN 0968-0896. http://www.sciencedirect.com/science/article/pii/S0968089616309099, DOI: 10.1016/j.bmc.2016.11.032. [COBISS.SI-ID 4248177]

12. KNEZ, Damijan, KOŠAK, Urban, BRUS, Boris, PIŠLAR, Anja, COQUELLE, Nicolas, STOJAN, Jure, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Structure-based drug design : from selective butyrylcholinesterase towards multifunctional anti-Alzheimer ligands. In: ANDERLUH, Gregor (ed.), PODOBNIK, Marjetka (ed.). Advances in structural biology : mini simpozij 2017 : [26th October 2017, Ljubljana]. Ljubljana: Department of Molecular Biology and Nanobiotechnology D11, National Institute of Chemistry, 2017. Str. 16, ilustr. ISBN 978-961-6104-37-1. [COBISS.SI-ID 4439921]

13. KNEZ, Damijan, COQUELLE, Nicolas, PIŠLAR, Anja, ŽAKELJ, Simon, JUKIČ, Marko, SOVA, Matej, MRAVLJAK, Janez, NACHON, Florian, BRAZZOLOTTO, Xavier, KOS, Janko, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Butyrylcholinesterase inhibitors grafted with antioxidant and neuroprotective activities : novel multifunctional ligands for Alzheimer's disease. In: 13th International Meeting on Cholinesterases and the 7th International Conference on Paraoxonases, Hradec Králové, Czech Republic 9 th - 14th September 2018. Hradec Králové: Univerzita obrany, Fakulta vojenského zdravotnictví, 2018. Str. 127. Military Medical Science Letters, Vol. 87, iss. 2, 2018. ISSN 2571-113X. https://www.mmsl.cz/artkey/mms-201802-0008_13th-international-meeting-on-cholinesterases-7th-international-conference-on-paraoxonases.php, http://system.bpp.cz/upload/files/Chepon2018/MMSL_2018_RGB_supplementum_1.pdf. [COBISS.SI-ID 4594289]

14. BRUS, Boris, KOŠAK, Urban, KNEZ, Damijan, COQUELLE, Nicolas, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Disubstituted piperidine derivatives as butyrylcholinesterase inhibitors for use in the treatment of Alzheimer : European patent specification EP 3256128 (B1), 2018-11-14. München: European Patent and Trademark Office, 2018. 47 str., ilustr. https://register.epo.org/application?number=EP16720556. [COBISS.SI-ID 4224113]
patent family: EP3256128 (A1), 2017-12-20; P201500076, 2015-03-25; US10071964 (B2), 2018-09-11; SI24951 (A), 2016-09-30; WO2016151484 (A1) , 2016-09-29

15. KOŠAK, Urban, BRUS, Boris, KNEZ, Damijan, ŽAKELJ, Simon, TRONTELJ, Jurij, PIŠLAR, Anja, ŠINK, Roman, JUKIČ, Marko, ŽIVIN, Marko, PODKOWA, Adrian, NACHON, Florian, BRAZZOLOTTO, Xavier, STOJAN, Jure, KOS, Janko, COQUELLE, Nicolas, SAŁAT, Kinga, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. The magic of crystal structure-based Inhibitor optimization : development of a butyrylcholinesterase inhibitor with picomolar affinity and In vivo activity. Journal of medicinal chemistry. 2018, vol. 61, iss. 1, str. 119-139, ilustr. ISSN 0022-2623. http://pubs.acs.org/doi/10.1021/acs.jmedchem.7b01086, DOI: 10.1021/acs.jmedchem.7b01086. [COBISS.SI-ID 4444017]

16. KNEZ, Damijan, COQUELLE, Nicolas, PIŠLAR, Anja, ŽAKELJ, Simon, JUKIČ, Marko, SOVA, Matej, MRAVLJAK, Janez, NACHON, Florian, BRAZZOLOTTO, Xavier, KOS, Janko, COLLETIER, Jacques-Philippe, GOBEC, Stanislav. Multi-target-directed ligands for treating Alzheimer's disease : butyrylcholinesterase inhibitors displaying antioxidant and neuroprotective activities. European journal of medicinal chemistry. [Print ed.]. Aug. 2018, vol. 156, str. 598-617, ilustr. ISSN 0223-5234. https://www.sciencedirect.com/science/article/pii/S0223523418305890, DOI: 10.1016/j.ejmech.2018.07.033. [COBISS.SI-ID 4547697]

17. PAJK, Stane, KNEZ, Damijan, KOŠAK, Urban, ZOROVIĆ, Maja, BRAZZOLOTTO, Xavier, COQUELLE, Nicolas, NACHON, Florian, COLLETIER, Jacques-Philippe, ŽIVIN, Marko, STOJAN, Jure, GOBEC, Stanislav. Development of potent reversible selective inhibitors of butyrylcholinesterase as fluorescent probes. Journal of enzyme inhibition and medicinal chemistry. 2020, vol. 35, iss. 1, str. 498-505, ilustr., graf. prikazi. ISSN 1475-6366. https://www.tandfonline.com/doi/full/10.1080/14756366.2019.1710502, Repozitorij Univerze v Ljubljani – RUL, DOI: 10.1080/14756366.2019.1710502. [COBISS.SI-ID 4869233]